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The Journal of Pain
Volume 12, Issue 3
, Pages 315-322
, March 2011
The Antinociceptive Effects of AR-A014418, a Selective Inhibitor of Glycogen Synthase Kinase-3 Beta, in Mice
References
- . Glycogen synthase kinase-3beta inhibition attenuates asthma in mice. Am J Respir Crit Care Med. 2007;176:431–438
- . Glutamate receptors and pain. Semin Cell Dev Biol. 2006;17:592–604
- . Structural insights and biological effects of glycogen synthase kinase 3-specific inhibitor AR-A014418. J Biol Chem. 2003;278:45937–45945
- . Glycogen synthase kinase 3 regulates N-methyl-D-aspartate receptor channel trafficking and function in cortical neurons. Mol Pharmacol. 2007;72:40–51
- . Antinociceptive mechanisms of orally administered decursinol in the mouse. Life Sci. 2003;73:471–485
- . Glycogen synthase kinase-3beta inhibition attenuates the development of bleomycin-induced lung injury. Int J Immunopathol Pharmacol. 2007;20:619–630
- . Glycogen synthase kinase-3beta inhibition attenuates the degree of arthritis caused by type II collagen in the mouse. Clin Immunol. 2006;120:57–67
- . Glycogen synthase kinase-3beta inhibitors protect against the organ injury and dysfunction caused by hemorrhage and resuscitation. Shock. 2006;25:485–491
- . Glycogen synthase kinase-3 from rabbit skeletal muscle. Separation from cyclic-AMP-dependent protein kinase and phosphorylase kinase. Eur J Biochem. 1980;107:519–527
- . GSK3 takes centre stage more than 20 years after its discovery. Biochem J. 2001;359:1–16
- . Contribution of spinal glutamatergic receptors to the antinociception caused by agmatine in mice. Brain Res. 2006;1093:116–122
- . CREB DNA binding activity is inhibited by glycogen synthase kinase-3 beta and facilitated by lithium. J Neurochem. 2001;78:1219–1232
- . Purification of glycogen synthase kinase 3 from rabbit skeletal muscle. Copurification with the activating factor (FA) of the (Mg-ATP) dependent protein phosphatase. Eur J Biochem. 1981;119:443–451
- . Formalin test in mice, a useful technique for evaluating mild analgesics. J Neurosci Methods. 1985;14:69–76
- . The formalin test in mice: Dissociation between inflammatory and non-inflammatory pain. Pain. 1987;30:103–114
- . Glycogen synthase kinase-3 (GSK3) in psychiatric diseases and therapeutic interventions. Curr Drug Targets. 2006;7:1421–1434
- . Glycogen synthase kinase-3 (GSK3): Inflammation, diseases, and therapeutics. Neurochem Res. 2007;32:577–595
- . Glycogen synthase kinase 3beta inhibitor Chir025 reduces neuronal death resulting from oxygen-glucose deprivation, glutamate excitotoxicity, and cerebral ischemia. Exp Neurol. 2004;188:378–386
- . The extent of cytokine induction in peripheral nerve lesions depends on the mode of injury and NMDA receptor signaling. J Neuroimmunol. 2004;149:77–83
- . Animal models of nociception. Pharmacol Rev. 2001;53:597–652
- . Toll-like receptor-mediated cytokine production is differentially regulated by glycogen synthase kinase 3. Nat Immunol. 2005;6:777–784
- . The induction of pain: An integrative review. Prog Neurobiol. 1999;57:161–164
- . Metabotropic glutamate receptors: Important modulators of nociception and pain behavior. Pain. 2002;98:1–8
- . Metabotropic glutamate receptors: Physiology, pharmacology, and disease. Annu Rev Pharmacol Toxicol. 2010;50:295–322
- . Effects of glycogen synthase kinase 3beta and cyclin-dependent kinase 5 inhibitors on morphine-induced analgesia and tolerance in rats. J Pharmacol Exp Ther. 2006;319:832–839
- . Cytokine-leukocyte networks and the establishment of pregnancy. Am J Reprod Immunol. 1997;37:438–442
- . Evidence for the involvement of glutamatergic system in the antinociceptive effect of ascorbic acid. Neurosci Lett. 2005;381:185–188
- . Glycogen synthase from rabbit skeletal muscle. Amino acid sequence at the sites phosphorylated by glycogen synthase kinase-3, and extension of the N-terminal sequence containing the site phosphorylated by phosphorylase kinase. Eur J Biochem. 1980;107:529–537
- . Contribution of interleukin-1 beta to the inflammation-induced increase in nerve growth factor levels and inflammatory hyperalgesia. Br J Pharmacol. 1995;115:1265–1275
- . Glycogen synthase kinase-3beta inhibits the xenobiotic and antioxidant cell response by direct phosphorylation and nuclear exclusion of the transcription factor Nrf2. J Biol Chem. 2006;281:14841–14851
- . Antinociceptive effect of meloxicam, in neurogenic and inflammatory nociceptive models in mice. Inflamm Res. 1998;47:302–307
- . Mechanisms involved in the antinociception caused by agmatine in mice. Neuropharmacology. 2005;48:1021–1034
- . Induction of nociceptive responses by intrathecal injection of interleukin-1 in mice. Life Sci. 1999;65:255–261
- . The formalin test: An evaluation of the method. Pain. 1992;51:5–17
- . IFN-beta production by TLR4-stimulated innate immune cells is negatively regulated by GSK3-beta. J Immunol. 2008;181:6797–6802
- . Reduction of experimental colitis in the rat by inhibitors of glycogen synthase kinase-3beta. Br J Pharmacol. 2006;147:575–582
- . Molecular cloning and expression of glycogen synthase kinase-3/factor A. EMBO J. 1990;9:2431–2438
- . Glycogen synthase kinase-3 regulates microglial migration, inflammation, and inflammation-induced neurotoxicity. Cell Signal. 2009;21:264–273
- . Ethical guidelines for investigations of experimental pain in conscious animals. Pain. 1983;16:109–110
Supported by grants from the Conselho Nacional de Desenvolvimento Científico e Tecnológico (CNPq), Fundação de Apoio à Pesquisa Científica Tecnológica do Estado de Santa Catarina (FAPESC), Financiadora de Estudos e Projetos (FINEP, Rede Instituto Brasileiro de Neurociência (IBN-Net, ref. 01.06.0842-00), Brazil), and the Spanish Ministry of Science and Innovation (Ref. SAF2006-08540 and Ref. PHB2007-0004-PC; Programa hispano-brasileño de cooperación interuniversitaria) awarded to M.G.L.
PII: S1526-5900(10)00581-X
doi: 10.1016/j.jpain.2010.06.007
© 2011 American Pain Society. Published by Elsevier Inc. All rights reserved.
« Previous
Next »
The Journal of Pain
Volume 12, Issue 3
, Pages 315-322
, March 2011
